Zeitschrift: ACS Medicinal Chemistry Letters

2022

Köhler, Leonhard ; Reich, Sebastian ; Yusenko, Maria ; Klempnauer, Karl-Heinz ; Shaikh, Amin H. ; Ahmed, Khursheed ; Begemann, Gerrit ; Schobert, Rainer ; Biersack, Bernhard:
A New Naphthopyran Derivative Combines c-Myb Inhibition, Microtubule-Targeting Effects, and Antiangiogenic Properties.
In: ACS Medicinal Chemistry Letters. Bd. 13 (2022) Heft 11 . - S. 1783-1790.
ISSN 1948-5875
DOI: https://doi.org/10.1021/acsmedchemlett.2c00403

2021

Fushimi, Makoto ; Buck, Hannes ; Balbach, Melanie ; Gorovyy, Anna ; Ferreira, Jacob ; Rossetti, Thomas ; Kaur, Navpreet ; Levin, Lonny R. ; Buck, Jochen ; Quast, Jonathan ; van den Heuvel, Joop ; Steegborn, Clemens ; Finkin-Groner, Efrat ; Kargman, Stacia ; Michino, Mayako ; Foley, Michael A. ; Miller, Michael ; Liverton, Nigel J. ; Huggins, David J. ; Meinke, Peter T.:
Discovery of TDI-10229 : A Potent and Orally Bioavailable Inhibitor of Soluble Adenylyl Cyclase (sAC, ADCY10).
In: ACS Medicinal Chemistry Letters. Bd. 12 (2021) Heft 8 . - S. 1283-1287.
ISSN 1948-5875
DOI: https://doi.org/10.1021/acsmedchemlett.1c00273

2020

Tomassi, Stefano ; Pfahler, Julian ; Mautone, Nicola ; Rovere, Anarita ; Esposito, Chiara ; Passeri, Daniela ; Pellicciari, Roberto ; Novellino, Ettore ; Pannek, Martin ; Steegborn, Clemens ; Paiardini, Alessandro ; Mai, Antonello ; Rotili, Dante:
From PARP1 to TNKS2 Inhibition : A Structure-Based Approach.
In: ACS Medicinal Chemistry Letters. Bd. 11 (2020) Heft 5 . - S. 862-868.
ISSN 1948-5875
DOI: https://doi.org/10.1021/acsmedchemlett.9b00654

You, Weijie ; Steegborn, Clemens:
Structural Basis for Activation of Human Sirtuin 6 by Fluvastatin.
In: ACS Medicinal Chemistry Letters. Bd. 11 (2020) Heft 11 . - S. 2285-2289.
ISSN 1948-5875
DOI: https://doi.org/10.1021/acsmedchemlett.0c00407